SCHEMBL11601593

SCHEMBL11601593

CCOC(=O)C(NC(=O)CCc1ccc([N+](=O)[O-])cc1)C(=O)OCC

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 1/20 0.48
KCNH2 Q12809 1/20 0.48
LMNA P02545 3/20 0.46
MAPT P10636 6/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
PKM P14618 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6776257 0.85 TRPV1 (0.53) LMNAMAPTKMT2AALDH1A1MEN1
SCHEMBL6782416 0.81 PPID (0.47) LMNAMAPTALDH1A1KDM4ECYP3A4
SCHEMBL20502747 0.80 ALDH1A1 (0.68) KMT2AALDH1A1PKM
SCHEMBL13991528 0.79 CYP4F2 (0.64) KCNJ1KCNH2LMNAMAPTKMT2A
SCHEMBL6781100 0.79 ALDH1A1 (0.45) LMNAMAPTALDH1A1KDM4E
SCHEMBL6774976 0.79 POLB (0.47) LMNAMAPTALDH1A1GAACYP2C19
SCHEMBL27541550 0.79 NAMPT (0.57) LMNAMAPTKMT2AALDH1A1MEN1
SCHEMBL7056969 0.78 KCNJ1 (0.54) KCNJ1KCNH2LMNAMAPTKMT2A
SCHEMBL7619439 0.78 ALDH1A1 (0.44) MAPTKMT2AALDH1A1MEN1KDM4E
SCHEMBL9386013 0.77 KMT2A (0.54) LMNAMAPTKMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4073929-A HYPOTENSIVE AGENTS MERCK & CO., INC. (US) 1978-02-14 US disclosed
US-4069333-A 2-HYDRAZINO-3-PHENYLPROPIONIC ACID DECARBOXYLASE INHIBITORS, BENZOXAZOLE ANALINES MERCK & CO., INC. (US) 1978-01-17 US disclosed
US-4051251-A DECARBOXYLASE INHIBITOR, BENZIMIDAZOLE AND BENZOXAZOLE ALANINES N MERCK & CO., INC. (US) 1977-09-27 US disclosed