SCHEMBL1161556

SCHEMBL1161556

Cn1c(CBr)nc2ccc(F)cc2c1=O

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.44
IDO2 Q6ZQW0 2/20 0.44
IDO1 P14902 1/20 0.44
HDAC6 Q9UBN7 1/20 0.42
CASR P41180 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
CASP3 P42574 2/20 0.40
PARP1 P09874 3/20 0.39
TNKS O95271 2/20 0.39
TNKS2 Q9H2K2 2/20 0.39
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
PARG Q86W56 1/20 0.39
HTR3A P46098 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1161773 0.88 HDAC6 (0.42) HDAC6CASRL3MBTL1KCNH2HRH3
SCHEMBL1161132 0.85 HDAC6 (0.45) TDO2IDO2IDO1HDAC6CASR
SCHEMBL1161602 0.83 L3MBTL1 (0.44) TDO2IDO2IDO1HDAC6CASR
SCHEMBL9919072 0.78 POLB (0.55) TDO2IDO2IDO1CASRL3MBTL1
SCHEMBL31542053 0.73 HDAC6 (0.56) HDAC6KCNH2
SCHEMBL5741522 0.72 USP2 (0.48) HDAC6CASP3PARG
SCHEMBL3820085 0.72 USP2 (0.47) HDAC6CASP3
SCHEMBL1161767 0.71 L3MBTL1 (0.44) HDAC6CASRL3MBTL1KCNH2HRH3
SCHEMBL16854205 0.70 HDAC1 (0.55) TDO2IDO2IDO1HDAC6L3MBTL1
SCHEMBL1161308 0.70 TRPV1 (0.41) HDAC6L3MBTL1POLBCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011012622-A1 BENZOXAZINONE DERIVATIVES FOR THE TREATMENT OF GLYTL MEDIATED DISORDERS GLAXO GROUP LIMITED (GB) 2011-02-03 WO disclosed
WO-2011012622-A1 BENZOXAZINONE DERIVATIVES FOR THE TREATMENT OF GLYTL MEDIATED DISORDERS GLAXO GROUP LIMITED (GB) 2011-02-03 WO disclosed