SCHEMBL1162028

SCHEMBL1162028

CCS(=O)(=O)Nc1cccc(N(Cc2ccc(Oc3cccc(OC4CCOC4)c3)cc2)c2ccccc2Cc2ccc(C#N)cc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 20/20 0.40
PGR P06401 2/20 0.35
NR3C2 P08235 2/20 0.35
AR P10275 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1162027 1.00 NR3C1 (0.40) NR3C1PGRNR3C2AR
SCHEMBL1162086 0.90 NR3C1 (0.48) NR3C1PGRNR3C2AR
SCHEMBL1161871 0.83 NR3C1 (0.57) NR3C1PGRNR3C2AR
SCHEMBL1161890 0.79 NR3C1 (0.51) NR3C1PGRNR3C2AR
SCHEMBL1161375 0.79 NR3C1 (0.59) NR3C1PGRNR3C2AR
SCHEMBL1161883 0.79 NR3C1 (0.61) NR3C1PGRNR3C2AR
SCHEMBL12015530 0.78 NR3C1 (0.48) NR3C1PGRNR3C2AR
SCHEMBL3969761 0.76 NR3C1 (0.69) NR3C1PGRNR3C2AR
SCHEMBL1161783 0.75 NR3C1 (0.51) NR3C1PGRNR3C2AR
SCHEMBL1161667 0.74 NR3C1 (0.45) NR3C1PGRNR3C2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2459524-A2 NOVEL COMPOUNDS AS MODULATORS OF GLUCOCORTICOID RECEPTORS Cadila Healthcare Limited (IN) 2012-06-06 EP disclosed
WO-2011016050-A2 NOVEL COMPOUNDS AS MODULATORS OF GLUCOCORTICOID RECEPTORS CADILA HEALTHCARE LIMITED (IN) 2011-02-10 WO disclosed