SCHEMBL11622285

SCHEMBL11622285

O=c1ccc(-c2ccc(Cl)c(C(F)(F)F)c2)n[nH]1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.68
NOTUM Q6P988 7/20 0.57
CYP1A2 P05177 3/20 0.57
PDE4A P27815 3/20 0.48
PDE4B Q07343 3/20 0.48
PDE4C Q08493 3/20 0.48
PDE4D Q08499 3/20 0.48
LMNA P02545 3/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
PDE3B Q13370 6/20 0.47
PDE3A Q14432 6/20 0.47
JAK2 O60674 1/20 0.44
NTRK1 P04629 1/20 0.44
RET P07949 1/20 0.44
PDGFRB P09619 1/20 0.44
CDK8 P49336 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44
AURKB Q96GD4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13070907 0.86 NOTUM (0.54) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL1769907 0.84 KDR (0.50) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL12649071 0.83 KDR (0.50) KDRNOTUMCYP1A2PDE4APDE4B
Potassium SCHEMBL11736530 0.83 LMNA (0.54) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL1769717 0.82 NOTUM (0.57) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL11622439 0.82 KDR (0.49) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL13071034 0.82 KDR (0.49) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL12648982 0.82 KDR (0.52) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL12595788 0.82 NOTUM (0.57) KDRNOTUMCYP1A2PDE4APDE4B
SCHEMBL3020961 0.81 LMNA (0.56) KDRNOTUMCYP1A2PDE4APDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4112095-A 6-Phenyl-1,2,4-triazolo[4,3-b]pyridazine hypotensive agents AMERICAN CYANAMID COMPANY (US) 1978-09-05 US disclosed