SCHEMBL11640488

SCHEMBL11640488

N#Cc1cc(C(O)CNC2CC2)cc(F)c1N

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.49
ADRB1 P08588 2/20 0.49
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
ADRB3 P13945 1/20 0.40
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11642580 0.95 ADRB2 (0.50) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11027251 0.95 ADRB2 (0.50) ADRB2ADRB1CYP1A2CYP3A4TSHR
Hydrochloric Acid SCHEMBL11042296 0.94 ADRB2 (0.49) ADRB2ADRB1CYP1A2CYP3A4TSHR
Hydrochloric Acid SCHEMBL11643322 0.89 ADRB2 (0.45) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11640814 0.85 ADRB2 (0.51) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11644150 0.85 ADRB2 (0.48) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11639398 0.85 ADRB2 (0.57) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11644239 0.85 ADRB2 (0.44) ADRB2ADRB1CYP1A2CYP3A4TSHR
SCHEMBL11641694 0.80 ADRB2 (0.53) ADRB2CYP1A2CYP3A4TSHRKDM4E
SCHEMBL11028356 0.80 ADRB2 (0.43) ADRB2ADRB1ADRB3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4119710-A ANALGESICS, UTEROSPASMOLYTICS, ANTISPASTICS, BLOCKING AGENTS BOEHRINGER INGELHEIM GMBH (DE) 1978-10-10 US disclosed