SCHEMBL11647201

SCHEMBL11647201

CCOC(=O)c1ccc(-c2ccccc2)nc1C(C(=O)O)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.51
MAPK1 P28482 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
MDM2 Q00987 2/20 0.49
CCR6 P51684 1/20 0.49
ALDH1A1 P00352 7/20 0.48
SMN1; SMN2 Q16637 6/20 0.48
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 2/20 0.48
MAPT P10636 4/20 0.48
LMNA P02545 2/20 0.48
ATM Q13315 2/20 0.48
TSHR P16473 2/20 0.47
TP53 P04637 1/20 0.47
GAA P10253 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4131672 0.82 KDM4E (0.54) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL4434197 0.82 MDM2 (0.67) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL29232726 0.81 CCR6 (0.56) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL8946445 0.81 MDM2 (0.68) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL9784691 0.81 KDM4E (0.55) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL4132138 0.77 MDM2 (0.60) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL28021689 0.75 PARP1 (0.62) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL28509330 0.74 MDM2 (0.60) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL31091350 0.74 MDM2 (0.60) KDM4EMAPK1TDP1L3MBTL1MDM2
SCHEMBL28516955 0.74 MDM2 (0.60) KDM4EMAPK1TDP1L3MBTL1MDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4117135-A NOVEL 5,6,7,8-TETRAHYDRO-5-QUINOLINES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS SCHERING, A.G. 1978-09-26 US disclosed