SCHEMBL11662986

SCHEMBL11662986

O=C1CNc2ncc(C(=O)O)cc2N1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
NNMT P40261 3/20 0.38
SMYD3 Q9H7B4 3/20 0.36
MB P02144 1/20 0.36
XIAP P98170 1/20 0.35
BIRC2 Q13490 1/20 0.35
MGAM O43451 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
GSK3A P49840 1/20 0.34
GSK3B P49841 1/20 0.34
CDK5 Q00535 1/20 0.34
CDK5R1 Q15078 1/20 0.34
CRBN Q96SW2 3/20 0.34
DDB1 Q16531 2/20 0.34
P4HA1 P13674 3/20 0.33
HCAR3 P49019 2/20 0.33
P4HTM Q9NXG6 2/20 0.33
MIF P14174 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14387476 0.83 MAP4K4 (0.42) HTTCYP11B1CYP11B2GSK3AGSK3B
SCHEMBL25789801 0.77 NNMT (0.49) NNMTMGAMP4HA1P4HTMMIF
SCHEMBL29712705 0.77 NNMT (0.49) NNMTMGAMP4HA1P4HTMMIF
SCHEMBL1255178 0.77 GSK3A (0.40) MBXIAPBIRC2CYP11B1CYP11B2
SCHEMBL16168388 0.77 NNMT (0.41) NNMTMGAMP4HA1P4HTMMIF
SCHEMBL28617969 0.76 NNMT (0.47) NNMTMGAMP4HA1P4HTMMIF
SCHEMBL16563482 0.76 AHR (0.39) MBXIAPBIRC2CYP11B1CYP11B2
SCHEMBL16564067 0.76 CYP11B1 (0.37) SMYD3MBXIAPBIRC2CYP11B1
SCHEMBL14387097 0.76 CYP11B1 (0.37) MBXIAPBIRC2CYP11B1CYP11B2
SCHEMBL1601643 0.76 CYP11B1 (0.37) MBXIAPBIRC2CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4091219-A ANTIINFLAMMATORY AGENTS, CNS DEPRESSANTS E. R. SQUIBB & SONS, INC. (US) 1978-05-23 US disclosed
US-4077955-A ANTIINFLAMMATORY, CNS DEPRESSANTS E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed