SCHEMBL11705115

SCHEMBL11705115

N#CC1(c2cccc(F)c2)CCCC(O)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 5/20 0.41
SLC6A4 P31645 4/20 0.41
KDM1A O60341 2/20 0.41
BDKRB1 P46663 1/20 0.38
ALDH1A1 P00352 2/20 0.36
CCR2 P41597 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
SLC6A2 P23975 1/20 0.35
TRPA1 O75762 1/20 0.34
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17985301 0.86 KDM1A (0.47) SLC6A3SLC6A4KDM1ABDKRB1ALDH1A1
SCHEMBL14491853 0.86 KDM1A (0.47) SLC6A3SLC6A4KDM1ABDKRB1ALDH1A1
SCHEMBL11706909 0.84 SLC6A3 (0.44) SLC6A3SLC6A4CCR2HTR2AHTR2C
SCHEMBL11704950 0.84 SLC6A3 (0.47) SLC6A3SLC6A4CCR2HTR2AHTR2C
SCHEMBL11704967 0.84 SLC6A3 (0.41) SLC6A3SLC6A4ALDH1A1SLC6A2KMT2A
SCHEMBL11703497 0.83 MEN1 (0.43) SLC6A3SLC6A4ALDH1A1KMT2ANPC1
SCHEMBL626449 0.81 KDM1A (0.43) SLC6A3SLC6A4KDM1ABDKRB1ALDH1A1
SCHEMBL1018956 0.81 SLC6A4 (0.46) SLC6A3SLC6A4KDM1ABDKRB1ALDH1A1
SCHEMBL1020648 0.79 SLC6A4 (0.49) SLC6A3SLC6A4KDM1ABDKRB1ALDH1A1
SCHEMBL11703241 0.79 SLC6A3 (0.40) SLC6A3SLC6A4ALDH1A1SLC6A2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4025558-A SPIRO(CYCLOHEXANE-1,1*(2'H)-NAPHTHALENE); BENZOSPIRAN DERIVATIVES; CNS DEPRESSANTS, LOWERS BLOOD PRESSURE THE UPJOHN COMPANY (US) 1977-05-24 US disclosed
US-4010201-A AMINOBENZOSPIRANS, CENTRAL NERVOUS SYSTEM DEPRESSANT, HYPOTENSIVE THE UPJOHN COMPANY (US) 1977-03-01 US disclosed
US-3932425-A CNS DEPRESSANT, BLOOD PRESSURE LOWERING THE UPJOHN COMPANY (US) 1976-01-13 US disclosed