SCHEMBL11708317

SCHEMBL11708317

O=C(c1ccc(F)cc1)C1CCN(CCn2c(=O)[nH]c3ccc(Cl)cc32)CC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.64
HTR2C P28335 4/20 0.64
CYP3A4 P08684 3/20 0.64
HPGD P15428 3/20 0.64
DRD2 P14416 3/20 0.64
HTR7 P34969 3/20 0.64
HTR6 P50406 3/20 0.64
ALDH1A1 P00352 2/20 0.64
CYP2C19 P33261 2/20 0.64
LMNA P02545 2/20 0.64
CYP1A2 P05177 2/20 0.64
HTR1A P08908 2/20 0.64
CYP2C9 P11712 2/20 0.64
MEN1 O00255 1/20 0.64
MAPT P10636 1/20 0.64
ADRA2B P18089 1/20 0.64
ADRA2C P18825 1/20 0.64
DRD1 P21728 1/20 0.64
DRD4 P21917 1/20 0.64
HTR1D P28221 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11713024 0.94 CYP3A4 (0.57) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL11708162 0.92 HTR2A (0.64) HTR2AHTR2CCYP3A4HPGDDRD2
Milenperone SCHEMBL29710910 0.87 CYP2D6 (0.58) HTR2AHTR2CCYP3A4HPGDDRD2
Milenperone SCHEMBL121986 0.87 CYP2D6 (0.58) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL8018901 0.86 HTR2A (0.78) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL11708157 0.83 HTR2A (0.58) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL11712014 0.83 HTR2A (0.57) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL11007280 0.80 HTR2A (0.81) HTR2AHTR2CCYP3A4HPGDDRD2
SCHEMBL11707541 0.80 HTR2A (0.69) HTR2AHTR2CCYP3A4HPGDDRD2
Declenperone SCHEMBL2112237 0.80 HTR2A (0.69) HTR2AHTR2CCYP3A4HPGDDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4035369-A 1-Benzazolylalkyl-4-substituted-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1977-07-12 US disclosed