SCHEMBL11712014

SCHEMBL11712014

Cc1ccc2[nH]c(=O)n(CCCN3CCC(C(=O)c4ccc(F)cc4)CC3)c2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.57
CYP3A4 P08684 3/20 0.57
CYP1A2 P05177 2/20 0.57
ALDH1A1 P00352 2/20 0.57
HPGD P15428 2/20 0.57
CYP2C19 P33261 2/20 0.57
LMNA P02545 2/20 0.57
KCNH2 Q12809 2/20 0.57
HTR2C P28335 2/20 0.57
HTR7 P34969 2/20 0.57
HTR6 P50406 2/20 0.57
MEN1 O00255 1/20 0.57
HTR1A P08908 1/20 0.57
MAPT P10636 1/20 0.57
CYP2C9 P11712 1/20 0.57
DRD2 P14416 1/20 0.57
ADRA2B P18089 1/20 0.57
ADRA2C P18825 1/20 0.57
DRD1 P21728 1/20 0.57
DRD4 P21917 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11707407 0.93 HTR2A (0.57) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL11707801 0.90 HTR2A (0.58) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL11713024 0.89 CYP3A4 (0.57) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
Declenperone SCHEMBL2112237 0.86 HTR2A (0.69) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL11708157 0.86 HTR2A (0.58) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL11707541 0.84 HTR2A (0.69) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL3404250 0.84 HTR2A (0.58) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
Milenperone SCHEMBL121986 0.83 CYP2D6 (0.58) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
Milenperone SCHEMBL29710910 0.83 CYP2D6 (0.58) HTR2ACYP3A4CYP1A2ALDH1A1HPGD
SCHEMBL11708317 0.83 HTR2A (0.64) HTR2ACYP3A4CYP1A2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4035369-A 1-Benzazolylalkyl-4-substituted-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1977-07-12 US disclosed