SCHEMBL11730100

SCHEMBL11730100

Cc1nnc2n1-c1ccccc1C(c1ccccc1F)=NC2

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTAFR P25105 7/20 0.76
GABRA1 P14867 8/20 0.71
GABRA5 P31644 8/20 0.71
GABRA2 P47869 8/20 0.71
GABRB2 P47870 7/20 0.71
BRD4 O60885 2/20 0.65
GABRA3 P34903 5/20 0.58
OPRK1 P41145 3/20 0.58
PDE4D Q08499 2/20 0.58
GABRG2 P18507 1/20 0.58
HTR2A P28223 1/20 0.58
GABRB3 P28472 1/20 0.58
ADRA1A P35348 1/20 0.58
TSHR P16473 1/20 0.56
HPGD P15428 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
LMNA P02545 1/20 0.53
CNR1 P21554 1/20 0.53
SLC22A1 O15245 1/20 0.49
ABCB11 O95342 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23881599 0.90 PTAFR (0.63) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL11620188 0.89 PTAFR (0.79) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL14282558 0.89 PTAFR (0.79) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL11858842 0.88 PTAFR (0.65) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL2841164 0.87 GABRA1 (0.76) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL11185785 0.87 PTAFR (0.76) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL7327360 0.87 GABRA1 (0.79) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL9378631 0.87 PTAFR (1.00) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL11395828 0.87 PTAFR (0.66) PTAFRGABRA1GABRA5GABRA2GABRB2
SCHEMBL29858197 0.87 GABRA1 (0.76) PTAFRGABRA1GABRA5GABRA2GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4018788-A 6-(O-Halophenyl)-1-methyl-4H-s-triazolo[4,3-a][1,4]-benzodiazepine THE UPJOHN COMPANY (US) 1977-04-19 US disclosed