SCHEMBL11733232

SCHEMBL11733232

S=C(Nc1nc2ccccc2[nH]1)c1cscn1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
LMNA P02545 2/20 0.49
NPC1 O15118 12/20 0.48
RAB9A P51151 10/20 0.48
SMN1; SMN2 Q16637 8/20 0.48
TP53 P04637 4/20 0.48
KDM4E B2RXH2 3/20 0.48
TDP1 Q9NUW8 2/20 0.48
CYP1A2 P05177 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
CYP2D6 P10635 1/20 0.48
TSHR P16473 1/20 0.48
CYP2C19 P33261 1/20 0.48
METAP2 P50579 1/20 0.48
METAP1 P53582 1/20 0.48
FKBP1A P62942 1/20 0.48
HIF1A Q16665 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL418792 0.84 NPC1 (0.60) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11734953 0.82 NPC1 (0.59) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11729485 0.79 LMNA (0.49) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11728204 0.79 LMNA (0.49) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11730127 0.78 LMNA (0.51) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11737313 0.77 NPC1 (0.51) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11732020 0.77 LMNA (0.50) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11730171 0.76 LMNA (0.49) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11734676 0.76 NPC1 (0.68) CYP3A4LMNANPC1RAB9ASMN1; SMN2
SCHEMBL11732709 0.74 NPC1 (0.50) CYP3A4LMNANPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4009164-A Novel 2-substituted-1,2,4-thiadiazole-[2,3-a]-benzimidazoles and process for their preparation SYNTEX (U.S.A.) INC. (US) 1977-02-22 US disclosed
US-3976654-A FUNGICIDE SYNTEX (U.S.A.) INC. (US) 1976-08-24 US disclosed
US-3946031-A FUNGICIDES SYNTEX INC. (US) 1976-03-23 US disclosed