SCHEMBL11735233

SCHEMBL11735233

COc1cc2c(cc1OC)C(C)(C)C(=O)N(CCCN(C)CCCN1C(=O)c3cc(OC)c(OC)cc3C(C)(C)C1=O)C2=O

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOB P27338 6/20 0.46
TDP1 Q9NUW8 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA1A P35348 1/20 0.40
ABCB1 P08183 1/20 0.40
SMPD1 P17405 3/20 0.38
BCHE P06276 1/20 0.37
ACHE P22303 1/20 0.37
TERT O14746 1/20 0.37
ALOX15 P16050 1/20 0.36
MAPT P10636 1/20 0.35
HCN4 Q9Y3Q4 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11535775 0.89 ABCB1 (0.56) CYP1A2CYP3A4ADRA2BADRA1AABCB1
SCHEMBL11738951 0.85 CYP1A2 (0.53) MAOBTDP1CYP1A2CYP3A4TSHR
SCHEMBL11816886 0.85 TDP1 (0.44) TDP1CYP1A2CYP3A4TSHRADRA2B
SCHEMBL11737033 0.84 TDP1 (0.56) MAOBTDP1CYP1A2CYP3A4TSHR
SCHEMBL11739860 0.84 TOP2A (0.46) TDP1CYP1A2CYP3A4TSHRADRA2B
SCHEMBL11734295 0.81 TDP1 (0.58) MAOBTDP1CYP1A2CYP3A4TSHR
SCHEMBL11738830 0.80 ABCB1 (0.53) TDP1CYP1A2CYP3A4ABCB1SMPD1
SCHEMBL11748982 0.79 ABCB1 (0.60) MAOBCYP1A2CYP3A4TSHRADRA2B
SCHEMBL11729888 0.78 MAOB (0.40) MAOBTDP1ACHETERTALOX15
SCHEMBL11735706 0.77 TDP1 (0.59) MAOBTDP1CYP1A2CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031219-A ANTIARRHYTHYMICS BOEHRINGER INGELHEIM GMBH (DT) 1977-06-21 US disclosed