SCHEMBL11738951

SCHEMBL11738951

COc1cc2c(cc1OC)C(C)(C)C(=O)N(CCN(C)CCN1C(=O)c3ccccc3C(C)(C)C1=O)C2=O

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
TSHR P16473 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA1A P35348 1/20 0.53
MAOB P27338 6/20 0.49
TDP1 Q9NUW8 1/20 0.47
PGR P06401 4/20 0.43
ALOX15 P16050 1/20 0.42
PARP1 P09874 1/20 0.41
ABCB1 P08183 1/20 0.41
HTR1A P08908 1/20 0.39
ADRA1B P35368 1/20 0.39
SMPD1 P17405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11737033 0.88 TDP1 (0.56) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11737697 0.87 MAOB (0.51) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11738968 0.87 TDP1 (0.64) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11735233 0.85 MAOB (0.46) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11735486 0.83 TDP1 (0.59) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11735706 0.83 TDP1 (0.59) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11741201 0.82 MAOB (0.47) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11748982 0.81 ABCB1 (0.60) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11738163 0.80 TDP1 (0.63) CYP1A2CYP3A4TSHRADRA2BADRA1A
SCHEMBL11734596 0.80 MAOB (0.53) CYP1A2CYP3A4TSHRADRA2BADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031219-A ANTIARRHYTHYMICS BOEHRINGER INGELHEIM GMBH (DT) 1977-06-21 US disclosed