SCHEMBL11749065

SCHEMBL11749065

COc1ccc([C@@H]2c3cc(OC)c(OC)cc3C[C@@H]3c4cc(OC)c(OC)cc4CCN23)cc1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
RAD52 P43351 1/20 0.52
DRD1 P21728 4/20 0.52
HTR1A P08908 1/20 0.52
TRPV1 Q8NER1 3/20 0.49
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
CA14 Q9ULX7 2/20 0.48
DRD2 P14416 3/20 0.48
KCNH2 Q12809 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11749061 1.00 MEN1 (0.53) MEN1KMT2ARAD52DRD1HTR1A
SCHEMBL11749707 0.84 DRD1 (0.56) KMT2ARAD52DRD1HTR1ADRD2
SCHEMBL11749701 0.84 DRD1 (0.56) KMT2ARAD52DRD1HTR1ADRD2
SCHEMBL16627026 0.80 DRD1 (0.53) DRD1TRPV1CA1CA2CA9
SCHEMBL16627024 0.80 DRD1 (0.53) DRD1TRPV1CA1CA2CA9
SCHEMBL11705438 0.78 GRIN2C (0.55) RAD52DRD1HTR1ADRD2KCNH2
SCHEMBL15610205 0.78 RAD52 (0.61) RAD52DRD1HTR1ADRD2
SCHEMBL14234700 0.78 RAD52 (0.61) RAD52DRD1HTR1ADRD2
SCHEMBL15610096 0.78 RAD52 (0.61) RAD52DRD1HTR1ADRD2
SCHEMBL9617443 0.78 RAD52 (0.61) RAD52DRD1HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4013666-A (8α,13Aβ)-8-CARBOCYCLIC/CARBOCYCLIC METHYL-5,8,13,13A-TETRAHYDRO-2,3,10,11-TETRAMETHOXY-6H-dibenzo[a,g]quinolizines and intermediates thereto G. D. SEARLE & CO. (US) 1977-03-22 US disclosed