SCHEMBL11750183

SCHEMBL11750183

CN1CCN(c2nsnc2OCC(O)CNC(C)(C)C)CC1

nearest known ligand 0.78

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 5/20 0.78
CYP2D6 P10635 4/20 0.78
ADRB1 P08588 4/20 0.78
HTR1A P08908 4/20 0.78
ADRB3 P13945 2/20 0.78
CYP1A2 P05177 2/20 0.78
DRD1 P21728 2/20 0.78
CYP3A4 P08684 1/20 0.78
NFKB1 P19838 1/20 0.78
SIGMAR1 Q99720 1/20 0.78
TDP1 Q9NUW8 1/20 0.78
SMN1; SMN2 Q16637 1/20 0.67
BLM P54132 1/20 0.67
ADRA2A P08913 3/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
ADRA1A P35348 2/20 0.42
RECQL P46063 1/20 0.42
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11750171 1.00 ADRB2 (0.78) ADRB2CYP2D6ADRB1HTR1AADRB3
SCHEMBL11405827 0.89 CYP2D6 (0.79) ADRB2CYP2D6ADRB1HTR1AADRB3
SCHEMBL11755099 0.89 CYP2D6 (0.79) ADRB2CYP2D6ADRB1HTR1AADRB3
Hydrochloric Acid SCHEMBL11418519 0.88 CYP2D6 (0.78) ADRB2CYP2D6ADRB1HTR1AADRB3
SCHEMBL11418535 0.87 ADRB2 (0.76) ADRB2CYP2D6ADRB1HTR1AADRB3
Timolol SCHEMBL222970 0.87 CYP1A2 (1.00) ADRB2CYP2D6ADRB1HTR1AADRB3
Timolol SCHEMBL2553603 0.87 CYP1A2 (1.00) ADRB2CYP2D6ADRB1HTR1AADRB3
Timolol SCHEMBL4912 0.87 CYP1A2 (1.00) ADRB2CYP2D6ADRB1HTR1AADRB3
Timolol SCHEMBL1587691 0.87 CYP1A2 (1.00) ADRB2CYP2D6ADRB1HTR1AADRB3
Timolol SCHEMBL7591293 0.86 CYP1A2 (0.98) ADRB2CYP2D6ADRB1HTR1AADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031125-A 3-Sulfonate ester of 2,3-dihydroxypropylamine MERCK & CO., INC. (US) 1977-06-21 US disclosed
US-3962338-A Novel methods and compounds employed therein MERCK & CO., INC. (US) 1976-06-08 US disclosed