SCHEMBL11752575

SCHEMBL11752575

O=C(c1ccc(Cl)cc1)C(Cl)c1ccc(Cl)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.50
CES1 P23141 3/20 0.50
TSHR P16473 2/20 0.48
ALOX15 P16050 1/20 0.48
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
MDM2 Q00987 3/20 0.44
BRD4 O60885 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
MAPK1 P28482 2/20 0.43
GSK3B P49841 2/20 0.43
SRD5A2 P31213 1/20 0.43
HIF1A Q16665 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
GAA P10253 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11751459 0.92 MAPK1 (0.57) CES2CES1TSHRALOX15CA1
SCHEMBL11750595 0.92 MAPK1 (0.57) CES2CES1TSHRALOX15CA1
SCHEMBL11755846 0.91 MDM2 (0.48) CES2CES1MDM2ALDH1A1LMNA
SCHEMBL11754522 0.91 MDM2 (0.48) CES2CES1MDM2ALDH1A1LMNA
SCHEMBL11754374 0.91 CES2 (0.58) CES2CES1TSHRMDM2MEN1
SCHEMBL11757043 0.91 MEN1 (0.44) CES2CES1TSHRALOX15CA1
SCHEMBL11755351 0.91 KMT2A (0.53) CES2CES1TSHRALOX15CA1
SCHEMBL11754114 0.91 KMT2A (0.53) CES2CES1TSHRALOX15CA1
SCHEMBL11746499 0.91 CES2 (0.58) CES2CES1TSHRMDM2MEN1
SCHEMBL11748763 0.91 MEN1 (0.44) CES2CES1TSHRALOX15CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4051250-A OXAZOLE, THIAZOLE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-27 US disclosed
US-3933840-A ANTIPHLOGISTIC MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-20 US disclosed