SCHEMBL11754342

SCHEMBL11754342

CC(S)C(=O)O.Fc1ccccc1-c1ncoc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 15/20 0.47
MAPK13 O15264 1/20 0.47
MAPK12 P53778 1/20 0.47
MAPK11 Q15759 1/20 0.47
ADORA2A P29274 1/20 0.42
LTB4R Q15722 1/20 0.38
CARM1 Q86X55 1/20 0.37
PTGS1 P23219 2/20 0.36
PTGS2 P35354 2/20 0.36
MEN1 O00255 1/20 0.36
FABP2 P12104 1/20 0.36
TSHR P16473 1/20 0.36
AKR1C4 P17516 1/20 0.36
ADRA2B P18089 1/20 0.36
CHRM3 P20309 1/20 0.36
HTR2C P28335 1/20 0.36
DRD3 P35462 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11750825 0.90 MAPK14 (0.41) MAPK14MAPK13MAPK12MAPK11ADORA2A
SCHEMBL11751581 0.85 MAPK14 (0.49) MAPK14ADORA2ACARM1MEN1KMT2A
SCHEMBL11751670 0.85 ADORA2A (0.42) MAPK14MAPK13MAPK12MAPK11ADORA2A
SCHEMBL11750246 0.85 MAPK14 (0.52) MAPK14ADORA2ALTB4RPTGS1PTGS2
SCHEMBL11752080 0.83 ALDH1A1 (0.45) MAPK14ADORA2AMEN1AKR1C3AKR1C2
SCHEMBL11749673 0.81 MAPK14 (0.53) MAPK14ADORA2ACARM1MEN1KMT2A
SCHEMBL11753979 0.80 MAPK14 (0.47) MAPK14ADORA2AMEN1KMT2A
SCHEMBL11749158 0.80 MAPK14 (0.47) MAPK14ADORA2AMEN1KMT2A
SCHEMBL11748061 0.79 MAPK14 (0.50) MAPK14ADORA2ACARM1MEN1KMT2A
SCHEMBL11752064 0.79 ADORA2A (0.55) MAPK14ADORA2ACARM1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4051250-A OXAZOLE, THIAZOLE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-27 US disclosed
US-3933840-A ANTIPHLOGISTIC MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1976-01-20 US disclosed