SCHEMBL11754569

SCHEMBL11754569

CC(C)NC[C@H](O)COc1nsnc1N1CCCCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 3/20 0.58
ADRB1 P08588 3/20 0.58
ADRB3 P13945 3/20 0.58
CYP2D6 P10635 2/20 0.58
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
HTR1A P08908 1/20 0.58
NFKB1 P19838 1/20 0.58
DRD1 P21728 1/20 0.58
SIGMAR1 Q99720 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SMN1; SMN2 Q16637 2/20 0.51
BLM P54132 1/20 0.51
LIPA P38571 6/20 0.47
LMNA P02545 2/20 0.45
HSD17B10 Q99714 2/20 0.45
ALDH1A1 P00352 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11755634 0.89 CYP1A2 (0.74) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11193337 0.89 CYP1A2 (0.74) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11405827 0.85 CYP2D6 (0.79) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11755099 0.85 CYP2D6 (0.79) ADRB2ADRB1ADRB3CYP2D6CYP1A2
Hydrochloric Acid SCHEMBL11418519 0.84 CYP2D6 (0.78) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11527669 0.83 LIPA (0.52) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL9854476 0.79 CYP1A2 (0.70) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL10983705 0.77 CYP1A2 (0.74) ADRB2ADRB1ADRB3CYP2D6CYP1A2
SCHEMBL11753911 0.77 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6MAPT
SCHEMBL11753904 0.77 ADRB2 (0.48) ADRB2ADRB1ADRB3CYP2D6MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4031125-A 3-Sulfonate ester of 2,3-dihydroxypropylamine MERCK & CO., INC. (US) 1977-06-21 US disclosed
US-3962338-A Novel methods and compounds employed therein MERCK & CO., INC. (US) 1976-06-08 US disclosed