SCHEMBL11765248

SCHEMBL11765248

CCOC(=O)C(C#N)=C(C)c1ccc(CC(C)C)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.43
MAPT P10636 2/20 0.39
ACACB O00763 1/20 0.38
LMNA P02545 4/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
USP2 O75604 1/20 0.37
CRHBP P24387 1/20 0.37
RAB9A P51151 1/20 0.37
CRHR2 Q13324 1/20 0.37
PTGS1 P23219 4/20 0.37
PTGS2 P35354 4/20 0.37
CYP2C9 P11712 2/20 0.37
AKR1C3 P42330 2/20 0.37
CXCR1 P25024 2/20 0.37
CXCR2 P25025 2/20 0.37
ALDH1A1 P00352 2/20 0.37
TSHR P16473 2/20 0.37
ALB P02768 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11783073 1.00 HPGD (0.43) HPGDMAPTACACBLMNAMEN1
SCHEMBL11138250 0.87 MAPT (0.46) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL11138252 0.87 MAPT (0.46) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL1553411 0.86 ALDH1A1 (0.42) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL1553412 0.86 ALDH1A1 (0.42) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL1554070 0.83 DHODH (0.44) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL1554071 0.83 DHODH (0.44) HPGDMAPTLMNAMEN1KMT2A
SCHEMBL11668967 0.82 PTGS1 (0.45) HPGDACACBLMNAMEN1KMT2A
SCHEMBL11639636 0.82 PTGS1 (0.45) HPGDACACBLMNAMEN1KMT2A
SCHEMBL1554675 0.81 MAPT (0.47) HPGDMAPTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-52118445-A None JP disclosed
JP-52062237-A None JP disclosed
JP-S52118445-A 2-CYANO-3-METHYL-3-(4-ISOBUTYLPHENYL)ACRYLIC ACID DERIVATIVES AND MET HOD OF PREPARING THE SAME GRELAN PHARMACEUT CO LTD 1977-10-04 JP disclosed
JP-S5262237-A PROCESS FOR PREPARATION OF ALPHA-SUBSTITUTED PHENYLALKANE CARBOXYLIC A CID ONO PHARMACEUT CO LTD 1977-05-23 JP disclosed