SCHEMBL11780985

SCHEMBL11780985

COC(=O)C1c2ccccc2N(C)c2ccc(Cl)cc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.52
HDAC7 Q8WUI4 1/20 0.52
HDAC5 Q9UQL6 1/20 0.52
PGR P06401 1/20 0.43
EGFR P00533 1/20 0.42
SRC P12931 1/20 0.42
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
GAA P10253 3/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11776203 0.92 HDAC4 (0.52) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL38661846 0.87 HDAC4 (0.67) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL2992029 0.87 HDAC4 (0.67) HDAC4HDAC7HDAC5EGFRSRC
SCHEMBL7702581 0.84 PGR (0.43) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL7702518 0.83 PGR (0.43) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL7703633 0.81 PGR (0.41) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL7702521 0.81 PGR (0.41) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL14564636 0.79 HDAC4 (0.45) HDAC4HDAC7HDAC5PGREGFR
SCHEMBL1981762 0.78 HDAC3 (0.44) HDAC4HDAC7HDAC5MEN1KMT2A
SCHEMBL3772600 0.78 HDAC4 (0.55) HDAC4HDAC7HDAC5EGFRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3979515-A THYMOANALEPTIC ACTIVITY ROUSSEL-UCLAF (FR) 1976-09-07 US disclosed
US-3957757-A THYMOANALEPTICS ROUSSEL-UCLAF (FR) 1976-05-18 US disclosed