SCHEMBL11782425

SCHEMBL11782425

CCOC(=O)COc1ccccc1C1C(C(=O)OC)=C(C)NC(C)=C1C(=O)OC

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 5/20 0.73
MAPT P10636 4/20 0.73
NR1I2 O75469 2/20 0.60
ADORA3 P0DMS8 3/20 0.57
CYP2C9 P11712 4/20 0.57
KDM4E B2RXH2 4/20 0.57
TP53 P04637 4/20 0.57
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 3/20 0.57
CYP2C19 P33261 3/20 0.57
KMT2A Q03164 3/20 0.57
HIF1A Q16665 3/20 0.57
HSD17B10 Q99714 3/20 0.57
TSHR P16473 3/20 0.57
MEN1 O00255 2/20 0.57
ALDH1A1 P00352 2/20 0.57
HPGD P15428 2/20 0.57
CYP2D6 P10635 2/20 0.57
NFKB1 P19838 2/20 0.57
THPO P40225 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11782443 0.96 GAA (0.68) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11782732 0.91 NR1I2 (0.64) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11780614 0.87 MAPT (0.61) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11782746 0.87 NR1I2 (0.59) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL7362882 0.86 NR1I2 (0.64) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11783778 0.85 GAA (0.55) GAAMAPTNR1I2CYP2C9TP53
SCHEMBL11780629 0.84 MAPT (0.57) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11784644 0.83 GAA (0.56) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL17371182 0.82 KDM4E (0.60) GAAMAPTNR1I2ADORA3CYP2C9
SCHEMBL11783784 0.81 GAA (0.52) GAAMAPTCYP2C9TP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3968117-A CARDIOVASCULAR BAYER AKTIENGESELLSCHAFT (DT) 1976-07-06 US disclosed
US-3959296-A CARDIOVASCULAR AGENTS BAYER AKTIENGESELLSCHAFT (DT) 1976-05-25 US disclosed