SCHEMBL7362882

SCHEMBL7362882

COC(=O)C1=C(C)NC(C)=C(C(=O)OC)C1c1ccccc1OCC(=O)O

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 2/20 0.64
KDM4E B2RXH2 5/20 0.58
GAA P10253 4/20 0.58
MAPT P10636 3/20 0.56
HSD17B10 Q99714 4/20 0.55
CYP2C9 P11712 4/20 0.55
ADORA3 P0DMS8 3/20 0.55
TP53 P04637 3/20 0.55
CYP1A2 P05177 3/20 0.55
CYP3A4 P08684 3/20 0.55
TSHR P16473 3/20 0.55
CYP2C19 P33261 3/20 0.55
KMT2A Q03164 3/20 0.55
HIF1A Q16665 3/20 0.55
CACNA1F O60840 3/20 0.55
CACNA1D Q01668 3/20 0.55
CACNA1S Q13698 3/20 0.55
CACNA1C Q13936 3/20 0.55
GMNN O75496 2/20 0.55
ABCB11 O95342 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11782732 0.90 NR1I2 (0.64) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL11782746 0.88 NR1I2 (0.59) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL11782425 0.86 GAA (0.73) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL10961715 0.86 KDM4E (0.62) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL11782443 0.85 GAA (0.68) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL29676206 0.84 NR1I2 (0.73) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL3034560 0.84 NR1I2 (0.73) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL7390505 0.83 MAPT (0.56) KDM4EMAPTHSD17B10TSHR
SCHEMBL11007706 0.83 KDM4E (0.59) NR1I2KDM4EGAAMAPTHSD17B10
SCHEMBL7414856 0.82 NR1I2 (0.67) NR1I2KDM4EGAAMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5378718-A Cardiovascular activity, hypotensive CEDONA PHARMACEUTICALS B.V. (NL) 1995-01-03 US disclosed
WO-1992002503-A1 NOVEL 1,4-DIHYDROPYRIDINE DERIVATIVES CEDONA PHARMACEUTICALS BV (NL) 1992-02-20 WO disclosed