SCHEMBL11787449

SCHEMBL11787449

NC(=O)C1C(=O)N(c2cccc([N+](=O)[O-])c2)C(=O)c2ccccc21

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 2/20 0.61
HPN P05981 1/20 0.47
TDP1 Q9NUW8 1/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
RECQL P46063 1/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
POLB P06746 1/20 0.42
CASP6 P55212 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
HIF1A Q16665 1/20 0.41
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11790251 0.90 SCN2A (0.62) SCN2AHPNTDP1MEN1KMT2A
SCHEMBL11791794 0.79 ALDH1A1 (0.55) MEN1KMT2ACA12CA2CA9
SCHEMBL11792049 0.78 HTT (0.43) MEN1KMT2ARECQLCYP2C19TSHR
SCHEMBL11791994 0.78 NOTUM (0.38) TDP1CA1CA2CA9POLB
SCHEMBL11669113 0.77 SCN2A (1.00) SCN2AHPNTDP1MEN1KMT2A
SCHEMBL30758587 0.77 SCN2A (1.00) SCN2AHPNTDP1MEN1KMT2A
SCHEMBL11787924 0.75 SCN2A (0.41) SCN2AMEN1KMT2ACA12CA1
SCHEMBL11792757 0.75 BRD4 (0.39) MEN1KMT2AL3MBTL1CYP1A2CYP3A4
SCHEMBL11787157 0.75 CA1 (0.37) SCN2AMEN1KMT2ACA12CA1
SCHEMBL11794014 0.74 SCN2A (0.40) SCN2AMEN1KMT2ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3998954-A 1,3(2H,4H)-Dioxoisoquinoline-4-carboxamides used as anti-inflammatory agents PFIZER INC. (US) 1976-12-21 US disclosed