SCHEMBL11794897

SCHEMBL11794897

COc1ccc2[nH]cc(C(=O)Cl)c2c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.74
MEN1 O00255 2/20 0.74
KMT2A Q03164 2/20 0.74
MAPT P10636 2/20 0.74
MITF O75030 1/20 0.74
RAB9A P51151 1/20 0.74
NPSR1 Q6W5P4 1/20 0.74
NR4A2 P43354 1/20 0.73
ALDH1A1 P00352 3/20 0.61
CYP1A2 P05177 2/20 0.61
CYP2C19 P33261 2/20 0.61
CYP2C9 P11712 1/20 0.61
CPT1A P50416 1/20 0.57
HTR4 Q13639 3/20 0.57
KDM4E B2RXH2 3/20 0.57
IMPDH2 P12268 1/20 0.55
IMPDH1 P20839 1/20 0.55
HSD17B10 Q99714 2/20 0.54
HPGD P15428 1/20 0.54
NPC1 O15118 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29950498 0.90 LMNA (0.64) LMNAMEN1KMT2AMAPTMITF
SCHEMBL7385581 0.88 LMNA (0.70) LMNAMEN1KMT2AMAPTMITF
SCHEMBL27273111 0.88 MAPT (0.74) LMNAMEN1KMT2AMAPTMITF
SCHEMBL27908679 0.87 NR4A2 (0.77) LMNAMEN1KMT2AMAPTMITF
SCHEMBL592889 0.87 NR4A2 (0.77) LMNAMEN1KMT2AMAPTMITF
SCHEMBL2834218 0.86 NR4A2 (0.75) LMNAMEN1KMT2AMAPTMITF
SCHEMBL8555897 0.85 LMNA (1.00) LMNAMEN1KMT2AMAPTMITF
SCHEMBL3633587 0.84 NR4A2 (0.73) LMNAMEN1KMT2AMAPTMITF
SCHEMBL5068806 0.84 NR4A2 (1.00) LMNAMEN1KMT2AMAPTMITF
SCHEMBL1558974 0.83 NR4A2 (0.71) LMNAMEN1KMT2AMAPTMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3980668-A Anti-arrhythimic 5-endo-(3-indolecarbonyloxy)-N-[amino-(lower)alkyl]bicyclo[2,2,1]heptane-2,3-di-endo-carboxylic acid imides BRISTOL-MYERS COMPANY (US) 1976-09-14 US disclosed
US-3980667-A Anti-arrhythmic 5-endo-substituted oxy-N-(aminoloweralkyl)bicycle [2.2.2.]oc BRISTOL-MYERS COMPANY (US) 1976-09-14 US disclosed