SCHEMBL11807441

SCHEMBL11807441

CCOC(=O)CN1C(=O)CN=C(c2ccccc2)c2cc(C(F)(F)F)ccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.57
MAPT P10636 5/20 0.57
NPSR1 Q6W5P4 4/20 0.54
NR1I2 O75469 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
OPRM1 P35372 1/20 0.52
OPRK1 P41145 1/20 0.52
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
RAB9A P51151 1/20 0.51
ATM Q13315 1/20 0.51
KDM4E B2RXH2 1/20 0.48
MCL1 Q07820 1/20 0.48
GAA P10253 1/20 0.47
HTT P42858 1/20 0.47
GPR55 Q9Y2T6 1/20 0.47
THRB P10828 1/20 0.47
PTGDR2 Q9Y5Y4 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11806409 0.90 TP53 (0.46) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL5352101 0.85 NPSR1 (0.69) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL5360020 0.85 SMN1; SMN2 (0.64) TP53MAPTNPSR1ALDH1A1SMN1; SMN2
SCHEMBL11804829 0.82 LMNA (0.63) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11576717 0.81 NPSR1 (0.59) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11580050 0.81 NPSR1 (0.58) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11812609 0.79 TP53 (0.52) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11578265 0.79 NPSR1 (0.56) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11578974 0.79 NPSR1 (0.56) TP53MAPTNPSR1NR1I2ADORA3
SCHEMBL11810202 0.79 PTGDR2 (0.53) TP53MAPTNPSR1NR1I2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3933816-A 3-(Substituted aminomethyl)-7-substituted-3,5-dihydro-as-triazino[4,3-a][1,5]benzodiazepines THE UPJOHN COMPANY (US) 1976-01-20 US disclosed