SCHEMBL11857052

SCHEMBL11857052

COC(=O)C(Cc1ccc(Cl)cc1Cl)c1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 5/20 0.55
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
L3MBTL1 Q9Y468 4/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
EPHX1 P07099 1/20 0.48
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GAA P10253 1/20 0.46
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3372127 0.92 L3MBTL1 (0.52) HDAC8CYP3A4CYP2C9KMT2AMEN1
SCHEMBL11861822 0.86 KMT2A (0.49) CYP3A4CYP2C9KMT2AMEN1CYP1A2
SCHEMBL11856270 0.85 CYP3A4 (0.48) HDAC8CYP3A4CYP2C9KMT2AMEN1
SCHEMBL6005346 0.84 HDAC8 (0.54) HDAC8CYP3A4CYP2C9KMT2AMEN1
SCHEMBL11857190 0.84 CYP3A4 (0.49) HDAC8CYP3A4CYP2C9KMT2AMEN1
SCHEMBL3371105 0.80 ESR1 (0.63) KMT2ACYP1A2CYP2D6CYP2C19L3MBTL1
SCHEMBL11850785 0.80 PPARG (0.44) HDAC8CYP3A4CYP2C9HTTALDH1A1
SCHEMBL22394846 0.80 CHRM1 (0.52) KMT2AMEN1L3MBTL1MAPK1HTT
SCHEMBL11857227 0.80 CYP3A4 (0.66) HDAC8CYP3A4CYP2C9KMT2AMEN1
SCHEMBL17513540 0.79 HDAC8 (0.47) HDAC8CYP3A4CYP2C9KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3991201-A 1-(β-Aryl-β-R-ethyl)imidazoles as antimicrobial agents JANSSEN PHARMACEUTICA N.V. (BE) 1976-11-09 US disclosed