SCHEMBL11861663

SCHEMBL11861663

c1ccc(-c2n[nH]c3c2Cc2ccccc2-3)nc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 5/20 0.66
CDK1 P06493 1/20 0.65
CDK2 P24941 1/20 0.65
CHEK1 O14757 2/20 0.58
PDGFRB P09619 2/20 0.50
LRRK2 Q5S007 2/20 0.46
HIF1A Q16665 3/20 0.43
PIM1 P11309 2/20 0.42
GSR P00390 1/20 0.42
MAPK8 P45983 2/20 0.41
MAPK9 P45984 2/20 0.41
NPC1 O15118 1/20 0.41
PLK4 O00444 1/20 0.41
DAPK3 O43293 1/20 0.41
PDGFRA P16234 1/20 0.41
LTK P29376 1/20 0.41
MAP2K2 P36507 1/20 0.41
FLT3 P36888 1/20 0.41
CSNK1A1 P48729 1/20 0.41
TDO2 P48775 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11861679 0.90 KDR (0.57) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL6968182 0.80 KDR (1.00) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL29819445 0.80 KDR (1.00) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL29644972 0.79 CDK1 (1.00) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL6969778 0.79 CDK1 (1.00) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL15311739 0.78 PDGFRB (0.58) KDRCDK1CDK2CHEK1PDGFRB
Hydrochloric Acid SCHEMBL15312449 0.77 PDGFRB (0.56) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL6968969 0.77 NPC1 (0.48) KDRCDK1CDK2CHEK1LRRK2
SCHEMBL6969359 0.75 KDR (0.74) KDRCDK1CDK2CHEK1PDGFRB
SCHEMBL11860279 0.75 KDR (0.64) KDRCDK1CDK2CHEK1PDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3932430-A Substituted indeno, naphtho and cyclohepta pyrazoles SANDOZ, INC. (US) 1976-01-13 US disclosed