SCHEMBL11862007

SCHEMBL11862007

Clc1ccc(-c2[nH]nc3c2Cc2cc4c(cc2-3)OCO4)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2K4 P45985 2/20 0.46
CHEK1 O14757 10/20 0.44
EIF2AK1 Q9BQI3 1/20 0.44
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA4 P22748 1/20 0.42
CA6 P23280 1/20 0.42
HIF1A Q16665 2/20 0.38
KDR P35968 1/20 0.37
PDGFRB P09619 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
NFKB1 P19838 1/20 0.37
CYP2C19 P33261 1/20 0.37
GRIA2 P42262 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11862001 0.90 CHEK1 (0.53) MAP2K4CHEK1EIF2AK1CA1CA2
SCHEMBL11865780 0.81 CHEK1 (0.53) CHEK1CA1CA2CA4CA6
SCHEMBL11864287 0.78 CHEK1 (0.65) CHEK1EIF2AK1PDGFRB
SCHEMBL11862375 0.77 CHEK1 (0.49) CHEK1KDRPDGFRB
SCHEMBL11865843 0.76 KDR (0.60) CHEK1KDRPDGFRB
SCHEMBL11842046 0.75 NPC1 (0.44) MAP2K4CHEK1EIF2AK1CA1CA2
SCHEMBL11863997 0.75 HIF1A (0.57) MAP2K4CHEK1HIF1AKDRMEN1
SCHEMBL11862289 0.74 CHEK1 (0.46) MAP2K4CHEK1
SCHEMBL11865766 0.73 CHEK1 (0.68) CHEK1KDRPDGFRB
SCHEMBL4044046 0.72 PDGFRB (0.44) MAP2K4EIF2AK1CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3932430-A Substituted indeno, naphtho and cyclohepta pyrazoles SANDOZ, INC. (US) 1976-01-13 US disclosed