SCHEMBL11869092

SCHEMBL11869092

NC(=O)c1nc(S)sc1N

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 1/20 0.38
DAPK3 O43293 1/20 0.32
CSNK1A1 P48729 1/20 0.32
LIMK1 P53667 1/20 0.32
TNK2 Q07912 1/20 0.32
ROCK1 Q13464 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
MAP2K3 P46734 2/20 0.31
IKBKB O14920 3/20 0.30
F2 P00734 1/20 0.30
HSP90AB1 P08238 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27886757 0.77 PDPK1 (0.40) PDPK1MAP2K3IKBKBF2
SCHEMBL26684112 0.74 PDPK1 (0.38) PDPK1MAP2K3IKBKBF2HSP90AB1
SCHEMBL12661719 0.74 PDPK1 (0.38) PDPK1DAPK3CSNK1A1LIMK1TNK2
SCHEMBL7264803 0.71 EEF2K (0.30)
SCHEMBL1477709 0.70 CCNA2 (0.41) PDPK1DAPK3CSNK1A1LIMK1TNK2
SCHEMBL13460071 0.69 PDPK1 (0.38) PDPK1IKBKBF2HSP90AB1
SCHEMBL18337153 0.69 LMNA (0.41) PDPK1LIMK1IKBKB
SCHEMBL6570704 0.68 PDPK1 (0.33) PDPK1IKBKB
SCHEMBL13460095 0.67 IKBKB (0.38) PDPK1IKBKB
SCHEMBL27957609 0.67 PDPK1 (0.36) PDPK1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024077391-A1 THIAZOLO[5,4-D]PYRIMIDINE COMPOUNDS, COMPOSITIONS COMPRISING THEM AND USES THEREOF UNIVERSITE DE MONTREAL (CA) 2024-04-18 WO disclosed
CN-103709119-B Preparation method of 5-aminothiazole-4-formamide SHANGHAI INST TECHNOLOGY 2015-05-20 CN disclosed
CN-103709119-A Preparation method of 5-aminothiazole-4-formamide SHANGHAI INST TECHNOLOGY 2014-04-09 CN disclosed
US-3993661-A Quinone methide photograhpic reagent precursors POLAROID CORPORATION (US) 1976-11-23 US disclosed