SCHEMBL1192011

SCHEMBL1192011

Cc1c(CC(=O)O)c2cc(F)ccc2n1Cc1ccc(S(=O)(=O)N2CCCC2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 17/20 0.61
PTGDR Q13258 5/20 0.59
LMNA P02545 2/20 0.59
CYP1A2 P05177 2/20 0.59
CYP3A4 P08684 2/20 0.59
CYP2C9 P11712 2/20 0.59
TSHR P16473 2/20 0.59
CYP2C19 P33261 2/20 0.59
PMP22 Q01453 2/20 0.59
KDM4E B2RXH2 1/20 0.59
BLM P54132 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59
MEN1 O00255 1/20 0.50
RGS12 O14924 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
PKM P14618 1/20 0.50
NFKB1 P19838 1/20 0.50
MAPK1 P28482 1/20 0.50
GNAI1 P63096 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1191035 0.98 PTGDR2 (0.61) PTGDR2PTGDRLMNACYP1A2CYP3A4
SCHEMBL1191881 0.92 PTGDR2 (0.66) PTGDR2PTGDRLMNACYP1A2CYP3A4
SCHEMBL1786345 0.84 PTGDR2 (0.74) PTGDR2
SCHEMBL1191888 0.80 PTGDR2 (0.69) PTGDR2PTGDRLMNACYP1A2CYP3A4
SCHEMBL1784633 0.77 PTGDR2 (0.63) PTGDR2
SCHEMBL1785920 0.76 PTGDR2 (0.62) PTGDR2
SCHEMBL3395183 0.76 PTGDR2 (0.68) PTGDR2PTGDRLMNACYP1A2CYP3A4
SCHEMBL5015665 0.75 PTGDR2 (0.75) PTGDR2
SCHEMBL1320560 0.74 LMNA (1.00) PTGDR2LMNACYP1A2CYP3A4CYP2C9
SCHEMBL6531234 0.74 PTGDR2 (1.00) PTGDR2PTGDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7888383-B2 Organic compounds NOVARTIS AG (CH) 2011-02-15 US disclosed
US-20090221578-A1 Organic Compounds NOVARTIS AG (CH) 2009-09-03 US disclosed
EP-1971574-A2 BICYCLIC HETEROCYCLIC COMPOUNDS AS ANTIINFLAMMATORY OR ANTIALLERGIC AGENTS Novartis AG (CH) 2008-09-24 EP disclosed
WO-2007065684-A2 BICYCLIC HETEROYCLIC COMPOUNDS AS ANTIINFLAMMATORY OR ANTIALLERGIC AGENTS NOVARTIS AG (CH) 2007-06-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221578-A1 Organic Compounds DRD4, RDX, DRD1 PTGDR2 618/4885PTGDR 151/4885LMNA 2662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.