Pyrrole

Pyrrole

SCHEMBL1194080

NC(=O)c1ccccn1.c1cc[nH]c1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.53
CES1 P23141 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.52
LMNA P02545 2/20 0.52
NAPRT Q6XQN6 1/20 0.52
P4HTM Q9NXG6 1/20 0.52
ALDH1A1 P00352 1/20 0.50
KMT2A Q03164 2/20 0.47
GSK3B P49841 1/20 0.46
MAPK1 P28482 1/20 0.45
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
MITF O75030 1/20 0.44
PKM P14618 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4914089 0.88 CES2 (0.67) CES2CES1L3MBTL1LMNANAPRT
SCHEMBL61183 0.88
SCHEMBL1505348 0.88
Hydrochloric Acid SCHEMBL17493405 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
SCHEMBL16143265 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
SCHEMBL9094627 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
Ammonia Solution, Strong SCHEMBL902138 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
SCHEMBL9064565 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
Hydrochloric Acid SCHEMBL1704886 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT
Hydrochloric Acid SCHEMBL30998088 0.86 CES2 (0.64) CES2CES1L3MBTL1LMNANAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 183 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029660-B P2X3And/or P2X2/3Compounds and methods 阿萨纳生物科技有限责任公司 2019-11-15 CN claimed
CN-110461854-A Process for preparing chiral 2, 3-dihydrothiazolo [3,2-A ] pyrimidin-4-ium compounds BASF SE 2019-11-15 CN claimed
CN-110267953-A Tetrahydroimidazo [4,5-C ] pyridine derivatives as inducers of PD-L1 internalization 因赛特公司 2019-09-20 CN claimed
CN-105814040-B The condensed 1,4- dihydro two of inhibitor as thermal excited transcryption factor 1 dislikes ene derivative 癌症研究科技有限公司 2019-07-30 CN claimed
CN-109952302-A Muscarine M1 receptor forward direction allosteric modulators 苏文生命科学有限公司 2019-06-28 CN claimed
CN-109890819-A Heterocyclic compound as immunomodulator 因赛特公司 2019-06-14 CN claimed
CN-104926801-B Substituted azetidine analog derivative, the pharmaceutical composition containing it and its application in antitumor 浙江大学 2019-06-04 CN claimed
CN-106164047-B 1,2- substituted cyclopentane as orexin receptor antagonists 武田药品工业株式会社 2019-04-16 CN claimed
CN-105209449-B Inhibitors of the kynurenine pathway 库拉德夫制药私人有限公司 2019-02-01 CN claimed
CN-106170486-B Novel indazolecarboxamides, method for the production thereof, pharmaceutical preparations containing the same and use thereof for producing medicaments 拜耳医药股份有限公司 2019-01-15 CN claimed
CN-107484415-A 1-cyanopyrrolidine compounds as USP30 inhibitors 特殊治疗有限公司 2017-12-15 CN claimed
CN-107231802-A Heterocyclic derivatives and use thereof 株式会社C&C新药研究所 2017-10-03 CN claimed
CN-103384668-B compounds and compositions for inhibition of NAMPT 福马TM有限责任公司 2017-05-31 CN claimed
CN-106458984-A 5, 6-disubstituted pyridine-2-carboxamides as cannabinoid receptor agonists 豪夫迈·罗氏有限公司 2017-02-22 CN claimed
CN-106456619-A Bicyclic heterocyclic derivatives as IRAK4 inhibitors 奥列基因发现技术有限公司 2017-02-22 CN claimed
CN-106456582-A TrkA kinase inhibitors, compositions and methods thereof 默沙东公司 2017-02-22 CN claimed
CN-104072480-B Quinolines and its preparation method and application 沈阳药科大学 2016-12-28 CN claimed
CN-103958473-B Amide compound, composition and application thereof ADVINUS THERAPEUTICS LTD. (IN) 2016-11-30 CN claimed
CN-106029660-A P2X 3 and/or P2X 2/3 compounds and methods 阿萨纳生物科技有限责任公司 2016-10-12 CN claimed
CN-103874686-B Piperidine derivatives and compositions for inhibition of nicotinamide phosphoribosyltransferase (NAMPT) 福马TM有限责任公司 2016-08-17 CN claimed