SCHEMBL11964652

SCHEMBL11964652

COc1ccc(CN2C(=O)C(Cc3ccccc3)N=C(Cl)c3cc(Cl)ccc32)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
ALDH2 P05091 1/20 0.46
ALDH3A1 P30838 1/20 0.46
SCN9A Q15858 1/20 0.42
CHRM5 P08912 2/20 0.42
TSHR P16473 1/20 0.41
BDKRB2 P30411 3/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
MMP1 P03956 1/20 0.41
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
CASP3 P42574 1/20 0.41
ATM Q13315 1/20 0.40
CES2 O00748 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12172272 0.95 CHRM5 (0.44) SCN9ACHRM5TSHRMAPT
SCHEMBL2117495 0.91 NPBWR1 (0.43) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL1515025 0.89 TSHR (0.43) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL1514972 0.89 TSHR (0.43) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL12099078 0.89 TSHR (0.43) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL10193349 0.89 CMA1 (0.44) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL10164821 0.87 CHRM5 (0.38) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL2119895 0.84 TSHR (0.42) ALDH1A1ALDH2ALDH3A1SCN9ACHRM5
SCHEMBL1515028 0.83 CHRM5 (0.39) ALDH1A1SCN9ACHRM5TSHRTP53
SCHEMBL1515068 0.83 CHRM5 (0.39) SCN9ACHRM5TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120289498-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2012-11-15 US disclosed
US-8242109-B2 Compositions and methods relating to novel compounds and targets thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2012-08-14 US disclosed
US-20110195959-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2011-08-11 US disclosed
US-7851465-B2 Compositions and methods relating to novel compounds and targets thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2010-12-14 US disclosed
US-20080269194-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2008-10-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080269194-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof BAX, BAD, BAK1 ALDH1A1 3248/4885ALDH2 912/4885ALDH3A1 3915/4885
US-20110195959-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof BAX, BAD, BAK1 ALDH1A1 3248/4885ALDH2 912/4885ALDH3A1 3915/4885
US-20120289498-A1 Compositions And Methods Relating To Novel Compounds And Targets Thereof BAX, BAD, BAK1 ALDH1A1 3248/4885ALDH2 912/4885ALDH3A1 3915/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.