SCHEMBL11967673

SCHEMBL11967673

COC(=O)CS(=O)(=O)N(Cc1ccc(CF)cc1)c1sc2ccccc2c1C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 5/20 0.50
PTPN1 P18031 4/20 0.37
PTPN6 P29350 1/20 0.37
PTPN11 Q06124 1/20 0.37
HSD11B1 P28845 1/20 0.37
MAPT P10636 3/20 0.37
TP53 P04637 2/20 0.36
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
CMA1 P23946 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1098460 0.88 TRPM8 (0.67) TRPM8
SCHEMBL1099222 0.83 TRPM8 (0.67) TRPM8TP53LMNA
SCHEMBL1098367 0.78 TRPM8 (0.65) TRPM8
SCHEMBL2060927 0.78 TRPM8 (0.40) TRPM8HSD11B1MAPTTP53KDM4E
SCHEMBL10280676 0.77 TRPM8 (0.71) TRPM8
SCHEMBL1107228 0.75 TRPM8 (0.66) TRPM8TP53HPGDNPSR1LMNA
SCHEMBL1098524 0.74 TRPM8 (0.64) TRPM8TP53LMNA
SCHEMBL1098599 0.73 TRPM8 (0.54) TRPM8TP53LMNA
SCHEMBL10280678 0.73 TRPM8 (0.46) TRPM8PTPN1HSD11B1MAPTTP53
SCHEMBL1099116 0.73 TRPM8 (0.69) TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2183239-B1 SULFONAMIDES AS TRPM8 MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2012-08-22 EP disclosed