SCHEMBL11977693

SCHEMBL11977693

Brc1c2ccccc2c(-c2ccc3c4ccccc4c4ccccc4c3c2)c2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.37
PTPN1 P18031 1/20 0.34
KDM4E B2RXH2 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HPRT1 P00492 3/20 0.32
MAPK1 P28482 2/20 0.32
MAPT P10636 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ALDH1A1 P00352 1/20 0.31
GRIN2D O15399 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3455378 0.86 GRIN2D (0.35) HPRT1MAPK1ALDH1A1GRIN2DGRIN2A
SCHEMBL17366608 0.86 ALDH1A1 (0.41) ALOX5KDM4EL3MBTL1HPGDHTT
SCHEMBL3000291 0.84 KDM4E (0.42) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL19283273 0.82 ALDH1A1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL17125452 0.82 ALDH1A1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL21517233 0.82 ALDH1A1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL276393 0.82 ALDH1A1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL2854881 0.82 ALDH1A1 (0.50) ALOX5CYP1A2HPGDCYP2C19HPRT1
SCHEMBL25625159 0.82 ALDH1A1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2
SCHEMBL14181764 0.81 PTPN1 (0.41) ALOX5PTPN1KDM4EL3MBTL1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2669262-B1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC CORP (JP) 2018-03-07 EP disclosed
EP-2669262-B1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC CORP (JP) 2018-03-07 EP disclosed
US-9070885-B2 Anthracene compound and organic electroluminescence element using same JNC CORPORATION (JP) 2015-06-30 US disclosed
US-9070885-B2 Anthracene compound and organic electroluminescence element using same JNC CORPORATION (JP) 2015-06-30 US disclosed
US-9070885-B2 Anthracene compound and organic electroluminescence element using same JNC CORPORATION (JP) 2015-06-30 US disclosed
EP-2669262-A1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC Corporation (JP) 2013-12-04 EP disclosed
US-20130292665-A1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC CORPORATION (JP) 2013-11-07 US disclosed
US-20130292665-A1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC CORPORATION (JP) 2013-11-07 US disclosed
US-20130292665-A1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC CORPORATION (JP) 2013-11-07 US disclosed
WO-2012102333-A1 NOVEL ANTHRACENE COMPOUND AND ORGANIC ELECTROLUMINESCENCE ELEMENT USING SAME JNC株式会社 (JP) 2012-08-02 WO disclosed