SCHEMBL11998124

SCHEMBL11998124

C#C[C@H]1CC[C@@H](C)N1C(=O)CNC1(C)CCN(c2cc(C(=O)O)ccn2)CC1

nearest known ligand 0.83

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 7/20 0.83
DPP8 Q6V1X1 1/20 0.64
DPP9 Q86TI2 1/20 0.64
PIK3CA P42336 2/20 0.41
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
KDM4C Q9H3R0 4/20 0.34
KDM5A P29375 2/20 0.34
KDM5B Q9UGL1 2/20 0.34
FFAR4 Q5NUL3 1/20 0.33
USP30 Q70CQ3 2/20 0.33
PTGER4 P35408 1/20 0.33
KDM6B O15054 1/20 0.33
KDM5C P41229 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
KDM4A O75164 1/20 0.33
MAPK14 Q16539 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14648444 0.95 DPP4 (0.92) DPP4DPP8DPP9PIK3CAKDM4C
SCHEMBL163502 0.91 DPP4 (1.00) DPP4DPP8DPP9PIK3CA
SCHEMBL2555136 0.91 DPP4 (1.00) DPP4DPP8DPP9PIK3CA
SCHEMBL882339 0.91 DPP4 (0.81) DPP4DPP8DPP9PIK3CAKDM4C
SCHEMBL20162036 0.91 DPP4 (1.00) DPP4DPP8DPP9PIK3CA
SCHEMBL646974 0.91 DPP4 (1.00) DPP4DPP8DPP9PIK3CA
SCHEMBL1040802 0.91 DPP4 (1.00) DPP4DPP8DPP9PIK3CA
SCHEMBL11997944 0.88 DPP4 (0.65) DPP4DPP8DPP9PDK1PDK2
SCHEMBL13287073 0.86 DPP4 (0.92) DPP4DPP8DPP9PIK3CA
SCHEMBL18175266 0.86 DPP4 (0.92) DPP4DPP8DPP9PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2057145-B1 SYNTHESIS OF (2S,5R)-5-ETHYNYL-1-{N-(4-METHYL-1-(4-CARBOXY-PYRIDIN-2-YL)PIPERIDIN-4-YL)GLYCYL}PYRROLIDINE-2-CARBONITRILE ABBOTT LAB (US) 2012-08-22 EP disclosed