SCHEMBL12016830

SCHEMBL12016830

CCOC(=O)c1c(C)c[nH]c1CCNCCCN1CCOCC1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 4/20 0.46
HSD17B10 Q99714 2/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
POLB P06746 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
RAD52 P43351 1/20 0.44
UHRF1 Q96T88 1/20 0.44
PAOX Q6QHF9 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.43
TP53 P04637 2/20 0.43
MAPT P10636 2/20 0.43
CYP3A4 P08684 1/20 0.42
MAPK1 P28482 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL155622 0.94 KDM4E (0.47) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL12016863 0.85 KDM4E (0.50) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL152626 0.84 KMT2A (0.40) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL2782550 0.83 ALDH1A1 (0.42) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL2782548 0.83 ALDH1A1 (0.42) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL2782588 0.83 ALDH1A1 (0.42) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL153614 0.83 ALDH1A1 (0.41) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL12017003 0.82 ALDH1A1 (0.40) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL150575 0.81 POLB (0.53) KDM4EALDH1A1HSD17B10GAAHPGD
SCHEMBL2780145 0.79 POLB (0.42) KDM4EALDH1A1HSD17B10GAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2179998-B1 2-(2-OXOINDOLINE-3-YLIDENE)METHYL-5-(2-HYDROXY-3-MORPHOLIN-4-YL -PROPYL)-6,7-DIHYDRO -1H- PYRROL[3,2-C]PYRIDINE-4(5H)-ONE COMPOUNDS AND USE AS PROTEIN KINASE INHIBITORS JIANGSU HENGRUI MEDICINE CO (CN) 2012-08-29 EP disclosed