SCHEMBL12021901

SCHEMBL12021901

CBc1ccc(C2=NCCCC2)cc1F

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 12/20 0.53
CHRNA3 P32297 12/20 0.53
CHRNA7 P36544 2/20 0.42
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
THRB P10828 1/20 0.34
CYP2C19 P33261 1/20 0.34
NISCH Q9Y2I1 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967805 0.76 CHRNB4 (0.57) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL29399603 0.71 CHRNB4 (0.50) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL206365 0.71 CHRNB4 (0.50) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL8151174 0.71 CHRNB4 (0.64) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL29396657 0.68 CHRNB4 (0.50) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL22097298 0.68 CHRNB4 (0.50) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL24233984 0.68 CHRNB4 (0.64) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL16098695 0.68 CHRNB4 (0.66) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL19253727 0.66 CHRNB4 (0.63) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2
SCHEMBL3935574 0.66 CHRNB4 (1.00) CHRNB4CHRNA3CHRNA7ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957477-B1 1H-BENZIMIDAZOLE-4-CARBOXAMIDES SUBSTITUTED WITH PHENYL AT THE 2-POSITION ARE POTENT PARP INHIBITORS ABBOTT LAB (US) 2011-12-07 EP disclosed