SCHEMBL1203062

SCHEMBL1203062

O=C(O)c1cnc2ccc(NCc3ccc(F)c(Cl)c3)nn12

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FYN P06241 4/20 0.60
IKBKB O14920 10/20 0.52
NTRK1 P04629 4/20 0.51
HDAC3 O15379 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC6 Q9UBN7 1/20 0.48
NTRK3 Q16288 1/20 0.47
NTRK2 Q16620 1/20 0.47
CHUK O15111 1/20 0.46
MAPK10 P53779 1/20 0.46
PIM1 P11309 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905622 0.90 FYN (0.72) FYNIKBKBNTRK1CHUKMAPK10
Hydrochloric Acid SCHEMBL1202037 0.89 FYN (0.71) FYNIKBKBNTRK1CHUKMAPK10
SCHEMBL2905868 0.87 FYN (0.50) FYNIKBKBNTRK1NTRK3NTRK2
SCHEMBL1202966 0.85 NTRK1 (0.50) FYNIKBKBNTRK1HDAC3HDAC1
SCHEMBL1203218 0.85 NTRK1 (0.49) FYNIKBKBNTRK1HDAC3HDAC1
SCHEMBL1202088 0.84 FYN (0.63) FYNNTRK1NTRK3NTRK2PIM1
SCHEMBL1203601 0.84 BRAF (0.51) FYNIKBKBNTRK1HDAC3HDAC1
SCHEMBL2905633 0.82 HDAC3 (0.46) FYNIKBKBHDAC3HDAC1HDAC2
SCHEMBL2902453 0.81 PIM1 (0.61) FYNIKBKBNTRK1NTRK3NTRK2
SCHEMBL1202134 0.81 IKBKB (0.65) FYNIKBKBNTRK1CHUKMAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110046127-A1 Imidazopyridazines for Use as Protein Kinase Inhibitors CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2011-02-24 US disclosed
EP-2217601-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2010-08-18 EP disclosed
WO-2009060197-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2009-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046127-A1 Imidazopyridazines for Use as Protein Kinase Inhibitors PIM1, PIM3, PIM2 FYN 403/4885IKBKB 297/4885NTRK1 755/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.