SCHEMBL2905622

SCHEMBL2905622

O=C(O)c1cnc2ccc(NCc3ccc(Cl)c(Cl)c3)nn12

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FYN P06241 2/20 0.72
IKBKB O14920 16/20 0.61
CHUK O15111 2/20 0.54
MAPK10 P53779 1/20 0.54
CDK2 P24941 1/20 0.51
NTRK1 P04629 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL1202037 0.99 FYN (0.71) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1203062 0.90 FYN (0.60) FYNIKBKBCHUKMAPK10NTRK1
SCHEMBL1202134 0.90 IKBKB (0.65) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1203467 0.87 IKBKB (0.76) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1202618 0.87 FYN (0.61) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1202657 0.86 FYN (0.72) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1202078 0.85 IKBKB (0.60) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL1203005 0.84 IKBKB (0.62) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL30521746 0.84 FYN (1.00) FYNIKBKBCHUKMAPK10CDK2
SCHEMBL2941291 0.84 FYN (1.00) FYNIKBKBCHUKMAPK10CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2217601-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS Centro Nacional de Investigaciones Oncológicas (CNIO) (ES) 2010-08-18 EP disclosed
WO-2009060197-A1 IMIDAZOPYRIDAZINES FOR USE AS PROTEIN KINASE INHIBITORS CENTRO NACIONAL DE INVESTIGACIONES ONCOLOGICAS (CNIO) (ES) 2009-05-14 WO disclosed