SCHEMBL12089979

SCHEMBL12089979

CC(C)(O)c1ccc(N2CCN(S(=O)(=O)c3ccc(Cl)nc3Cl)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.50
GCK P35557 8/20 0.46
GCKR Q14397 2/20 0.46
MAPT P10636 4/20 0.43
MEN1 O00255 2/20 0.43
LMNA P02545 2/20 0.43
KMT2A Q03164 2/20 0.43
ACLY P53396 1/20 0.42
TP53 P04637 2/20 0.41
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17467 0.87 GCK (0.61) HSD11B1GCKGCKRMAPTMEN1
SCHEMBL12089978 0.81 GCK (0.53) HSD11B1GCKGCKRMEN1KMT2A
SCHEMBL12089907 0.81 HSD11B1 (0.50) HSD11B1GCKGCKRMAPTMEN1
SCHEMBL12089425 0.80 GCK (0.57) HSD11B1GCKGCKRMAPTMEN1
SCHEMBL15200964 0.79 GCK (0.65) HSD11B1GCKGCKR
SCHEMBL12089435 0.75 GCK (0.57) HSD11B1GCKGCKRMAPTMEN1
SCHEMBL12088782 0.75 GCK (0.72) HSD11B1GCKMAPTMEN1LMNA
SCHEMBL25230194 0.74 POLB (0.47) MAPTMEN1LMNAKMT2ATSHR
SCHEMBL30466353 0.74 POLB (0.47) MAPTMEN1LMNAKMT2ATSHR
SCHEMBL12089376 0.74 GCK (0.54) HSD11B1GCKGCKRMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8431563-B2 Compounds that interact with glucokinase regulatory protein for the treatment of diabetes AMGEN INC. (US) 2013-04-30 US disclosed
US-20120225854-A1 COMPOUNDS THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES AMGEN INC. (US) 2012-09-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120225854-A1 COMPOUNDS THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES GCKR, GCK, SLC5A2 HSD11B1 1443/4885GCK 2/4885GCKR 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.