Udenafil

Udenafil

SCHEMBL120993

CCCOc1ccc(S(=O)(=O)NCCC2CCCN2C)cc1-c1nc2c(CCC)nn(C)c2c(=O)[nH]1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PDE5A

The experimentally established mechanism targets of Udenafil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE5A known ✓ O76074 19/20 1.00
PDE2A O00408 1/20 0.64
PDE9A O76083 1/20 0.64
PDE4A P27815 1/20 0.64
PDE6C P51160 1/20 0.64
PDE1A P54750 1/20 0.64
PDE11A Q9HCR9 1/20 0.64
PDE10A Q9Y233 1/20 0.64
KDM4E B2RXH2 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Udenafil SCHEMBL30452348 1.00 PDE5A (1.00) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8054822 0.97 PDE5A (0.94) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055636 0.97 PDE5A (0.94) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055433 0.97 PDE5A (0.94) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055565 0.95 PDE5A (0.91) PDE5APDE2APDE9APDE4APDE6C
SCHEMBL16850578 0.95 PDE5A (0.91) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055012 0.94 PDE5A (0.89) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055765 0.94 PDE5A (0.89) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8066232 0.94 PDE5A (0.89) PDE5APDE2APDE9APDE4APDE6C
Udenafil SCHEMBL8055102 0.94 PDE5A (0.89) PDE5APDE2APDE9APDE4APDE6C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 920 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12465605-B2 Methods and materials for gender-dependent treatment of cardiovascular dysfunction MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH (US) 2025-11-11 US claimed
US-20210060123-A1 THERAPEUTIC USE OF P75NTR NEUROTROPHIN BINDING PROTEIN LEVICEPT LTD (GB) 2021-03-04 US claimed
US-20180161392-A1 THERAPEUTIC USE OF P75NTR NEUROTROPHIN BINDING PROTEIN LEVICEPT LTD (GB) 2018-06-14 US claimed
US-20170231931-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES FUNDACIÓN PARA LA INVESTIGACIÓN MÉDICA APLICADA (ES) 2017-08-17 US claimed
EP-2825208-B1 P75NTR NEUROTROPHIN BINDING PROTEIN FOR THERAPEUTIC USE LEVICEPT LTD (GB) 2017-05-17 EP claimed
US-20150037335-A1 THERAPEUTIC USE OF P75NTR NEUROTROPHIN BINDING PROTEIN LEVICEPT LTD (GB) 2015-02-05 US claimed
EP-2825208-A1 THERAPEUTIC USE OF P75NTR NEUROTROPHIN BINDING PROTEIN Levicept Ltd. (GB) 2015-01-21 EP claimed
EP-2175728-B1 SODIUM CHANNEL INHIBITORS ICAGEN INC (US) 2014-09-10 EP claimed
WO-2013136078-A1 THERAPEUTIC USE OF P75NTR NEUROTROPHIN BINDING PROTEIN LEVICEPT LTD (GB) 2013-09-19 WO claimed
US-20090111837-A1 USE OF PDE7 INHIBITORS FOR THE TREATMENT OF NEUROPATHIC PAIN PFIZER INC. 2009-04-30 US claimed
WO-2007072169-A2 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF LUTS COMPRISING A PDE5 INHIBITOR AND A MUSCARINIC ANTAGONIST PFIZER PRODUCTS INC. (US) 2007-06-28 WO claimed
JP-2006528229-A 2006-12-14 JP claimed
WO-2006092691-A1 USE OF PDE7 INHIBITORS FOR THE TREATMENT OF NEUROPATHIC PAIN PFIZER LIMITED (GB) 2006-09-08 WO claimed
US-20060148693-A1 Composition comprising a pulmonary surfactant and a pde5 inhibitor for the treatment of lung diseases ALTANA PHARMA AG (DE) 2006-07-06 US claimed
US-20060094723-A1 Composition comprising a pde4 inhibitor and a pde5 inhibitor NYCOMED GMBH (DE) 2006-05-04 US claimed
EP-1638567-A1 COMPOSITION COMPRISING A PULMONARY SURFACTANT AND A PDE5 INHIBITOR FOR THE TREATMENT OF LUNG DISEASES ALTANA Pharma AG (DE) 2006-03-29 EP claimed
EP-1628682-A2 COMPOSITION COMPRISING A PDE4 INHIBITOR AND A PDE5 INHIBITOR ALTANA Pharma AG (DE) 2006-03-01 EP claimed
WO-2004110450-A1 COMPOSITION COMPRISING A PULMONARY SURFACTANT AND A PDE5 INHIBITOR FOR THE TREATMENT OF LUNG DISEASES ALTANA PHARMA AG (DE) 2004-12-23 WO claimed
WO-2004103407-A2 COMPOSITION COMPRISING A PDE4 INHIBITOR AND A PDE5 INHIBITOR ALTANA PHARMA AG (DE) 2004-12-02 WO claimed
US-20040132731-A1 Novel combination PFIZER, INC. 2004-07-08 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170231931-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES SNCA, PSEN2, PSEN1 PDE5A 545/4885PDE2A 540/4885PDE9A 2785/4885
US-20060094723-A1 Composition comprising a pde4 inhibitor and a pde5 inhibitor PDE5A, PDE12, PDE4A PDE5A 1/4885PDE2A 8/4885PDE9A 10/4885
US-20090111837-A1 USE OF PDE7 INHIBITORS FOR THE TREATMENT OF NEUROPATHIC PAIN PDE7A, PDE7B, PDE3A PDE5A 5/4885PDE2A 6/4885PDE9A 13/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.