Trestolone Acetate

Trestolone Acetate

SCHEMBL12101463

CC(=O)O[C@H]1CCC2C3C(CC[C@@]21C)C1CCC(=O)C=C1C[C@H]3C

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 7/20 0.70
MAPT P10636 2/20 0.55
LMNA P02545 2/20 0.55
PGR P06401 6/20 0.52
NR3C2 P08235 2/20 0.52
SERPINA6 P08185 2/20 0.50
ALDH1A1 P00352 2/20 0.47
SHBG P04278 2/20 0.47
SLC22A1 O15245 1/20 0.47
THRB P10828 1/20 0.47
MCL1 Q07820 1/20 0.47
CYP1A2 P05177 1/20 0.47
HIF1A Q16665 1/20 0.47
HSD17B10 Q99714 1/20 0.47
ESR1 P03372 2/20 0.45
MEN1 O00255 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
MAPK1 P28482 1/20 0.45
BRCA1 P38398 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trestolone Acetate SCHEMBL17302787 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL17302820 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL7779251 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL2787569 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL25863451 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL17302814 1.00 AR (0.70) ARMAPTLMNAPGRNR3C2
Trestolone Acetate SCHEMBL28108545 0.96 AR (0.65) ARMAPTLMNAPGRNR3C2
SCHEMBL24102452 0.92 AR (0.70) ARMAPTLMNAPGRNR3C2
SCHEMBL24102904 0.91 AR (0.69) ARMAPTLMNAPGRNR3C2
SCHEMBL24102896 0.91 AR (0.69) ARMAPTLMNAPGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230227492-A1 MONOMERIC AND OLIGOMERIC COMPOUND EMBODIMENTS AS CONTRACEPTIVES AND THERAPIES AND METHODS OF MAKING AND USING THE SAME THE USA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2023-07-20 US disclosed
EP-1608670-B1 PROCESS FOR THE PRODUCTION OF TIBOLONE RESOLUTION CHEMICALS LTD (GB) 2013-09-11 EP disclosed
EP-2497776-A2 Process for the production of tibolone Resolution Chemicals Limited (GB) 2012-09-12 EP disclosed
US-7884222-B2 protecting the 17-hydroxy group and the 3-keto group of nandrolone, then halogenating, methylating, isomerizing, dehydrogenating, reducing, oxidizing, ethynylating and deprotecting to form 17 beta -hydroxy-7 alpha -methyl-19-nor-17 alpha -pregn-5(10)-ene-20-yne-3-one RESOLUTION CHEMICALS LIMITED (GB) 2011-02-08 US disclosed
US-7884222-B2 protecting the 17-hydroxy group and the 3-keto group of nandrolone, then halogenating, methylating, isomerizing, dehydrogenating, reducing, oxidizing, ethynylating and deprotecting to form 17 beta -hydroxy-7 alpha -methyl-19-nor-17 alpha -pregn-5(10)-ene-20-yne-3-one RESOLUTION CHEMICALS LIMITED (GB) 2011-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230227492-A1 MONOMERIC AND OLIGOMERIC COMPOUND EMBODIMENTS AS CONTRACEPTIVES AND THERAPIES AND METHODS OF MAKING AND USING THE SAME SHBG, CYP19A1, GNRHR AR 7/4885MAPT 4428/4885LMNA 388/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.