SCHEMBL12101596

SCHEMBL12101596

Bc1ccc2c(O)c(C(=O)NCC(=O)OC(C)(C)C)c(=O)n(C)c2n1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 2/20 0.46
HIF1A Q16665 16/20 0.45
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2578845 0.89 EGLN1 (0.51) EGLN1HIF1AMEN1NPC1RAB9A
SCHEMBL2576963 0.86 HIF1A (0.48) EGLN1HIF1AMEN1NPC1RAB9A
SCHEMBL12101654 0.85 EGLN1 (0.58) EGLN1HIF1A
SCHEMBL2577063 0.85 HIF1A (0.44) EGLN1HIF1A
SCHEMBL12172226 0.84 EGLN1 (0.43) EGLN1HIF1ARAB9AKMT2AKDM4E
SCHEMBL2582034 0.84 HIF1A (0.48) EGLN1HIF1AMEN1NPC1RAB9A
SCHEMBL337546 0.82 EGLN1 (0.50) EGLN1HIF1AMEN1NPC1RAB9A
SCHEMBL2587881 0.82 CALCA (0.42) EGLN1HIF1AKDM4E
SCHEMBL2580935 0.82 EGLN1 (0.42) EGLN1HIF1A
SCHEMBL337574 0.80 EGLN1 (0.49) EGLN1HIF1AMEN1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097416-B1 AZAQUINOLONE BASED COMPOUNDS EXHIBITING PROLYL HYDROXYLASE INHIBITORY ACTIVITY, COMPOSITIONS, AND USES THEREOF AMGEN INC (US) 2012-09-12 EP disclosed