SCHEMBL12101652

SCHEMBL12101652

C=C(C)/N=C\N(N)c1ncc(OC)c2c(C(=O)C(=O)O)c[nH]c12

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.39
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
KCNH2 Q12809 1/20 0.35
MITF O75030 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12101629 0.91 CYP2C9 (0.36) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL9914969 0.82 CYP2C9 (0.41) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL9914931 0.82 CYP2C9 (0.47) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL9914927 0.80 CYP2C9 (0.45) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL9914923 0.77 CYP2C9 (0.43) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL14385656 0.77 CYP2C9 (0.48) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL12513521 0.75 CYP2C9 (0.45) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL10326156 0.74 CYP2C9 (0.38) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL12238398 0.74 CYP2C9 (0.47) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6
SCHEMBL10326256 0.74 CYP2C9 (0.47) CYP2C9CYP3A4CYP1A2CYP2C8CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2497770-A1 Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives Bristol-Myers Squibb Company (US) 2012-09-12 EP disclosed