SCHEMBL14385656

SCHEMBL14385656

C=C(C)/N=C\N(N)c1ncc(OC)c2c(C(=O)C(=O)N3CCN(c4nccn4-c4ccccc4)CC3)c[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.48
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C8 P10632 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
KCNH2 Q12809 1/20 0.43
DPP4 P27487 1/20 0.34
MAPT P10636 1/20 0.33
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14385717 0.84 CYP2C9 (0.44) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL12513521 0.80 CYP2C9 (0.45) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL9914931 0.80 CYP2C9 (0.47) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL9914927 0.78 CYP2C9 (0.45) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL13116907 0.78 CYP2C9 (0.72) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL12101652 0.77 CYP2C9 (0.39) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL14386385 0.77 CYP2C9 (0.40) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL9914923 0.76 CYP2C9 (0.43) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL15494335 0.75 CYP2C9 (0.46) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8
SCHEMBL12101629 0.74 CYP2C9 (0.36) CYP2C9CYP3A4CYP2D6CYP1A2CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007127635-A2 DIKETO-PIPERAZINE AND PIPERIDINE DERIVATIVES AS ANTIVIRAL AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-11-08 WO disclosed