SCHEMBL12101994

SCHEMBL12101994

CCn1c(=O)c(C)cc2c(C)nc(Nc3ccc(F)cc3)nc21

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 5/20 0.52
CCND1 P24385 5/20 0.52
CCND2 P30279 5/20 0.52
CCND3 P30281 5/20 0.52
ALDH1A1 P00352 2/20 0.51
HSD17B10 Q99714 2/20 0.51
KDM4E B2RXH2 2/20 0.51
GLA P06280 1/20 0.51
GAA P10253 1/20 0.51
HPGD P15428 1/20 0.51
MAPK1 P28482 1/20 0.51
HTT P42858 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
USP2 O75604 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
PIK3CA P42336 2/20 0.39
KCNH3 Q9ULD8 2/20 0.39
PIK3CD O00329 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL189479 0.90 ALDH1A1 (0.66) CDK4CCND1CCND2CCND3ALDH1A1
SCHEMBL189237 0.78 HSD17B10 (0.69) CDK4CCND1CCND2CCND3ALDH1A1
SCHEMBL189165 0.77 FGFR1 (0.51) CDK4CCND1CCND2CCND3ALDH1A1
SCHEMBL189369 0.76 ALDH1A1 (0.63) ALDH1A1HSD17B10KDM4EGLAGAA
SCHEMBL188479 0.75 WEE1 (0.45) CDK4CCND1CCND2CCND3ALDH1A1
SCHEMBL189950 0.75 RIPK2 (0.49) CDK4CCND1CCND2CCND3ALDH1A1
SCHEMBL189050 0.73 WEE1 (0.47) CDK4CCND1CCND3SRCCCNA2
SCHEMBL188663 0.73 ALDH1A1 (0.65) ALDH1A1HSD17B10KDM4EGLAGAA
SCHEMBL2632910 0.73 PIK3CA (0.50) ALDH1A1HSD17B10KDM4EGLAGAA
SCHEMBL3339784 0.73 KDM4E (0.58) CDK4CCND1CCND2CCND3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1931670-B1 PYRIDOPYRIMIDINONE INHIBITORS OF PI3K EXELIXIS INC (US) 2012-09-12 EP disclosed