SCHEMBL12102198

SCHEMBL12102198

CC(C)NC(=O)NCCOc1ccc2c(c1)C(C1(c3ccc(N)cc3)CCC1)NCC2

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.56
CYP3A4 P08684 1/20 0.56
MTNR1A P48039 7/20 0.34
MTNR1B P49286 7/20 0.34
NQO2 P16083 5/20 0.34
KDM4E B2RXH2 2/20 0.34
POLB P06746 1/20 0.34
ABCB1 P08183 1/20 0.34
HRH3 Q9Y5N1 3/20 0.32
HTR1A P08908 1/20 0.32
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
ACHE P22303 1/20 0.32
PPARG P37231 1/20 0.32
PPARD Q03181 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8016298 0.92 SLC6A9 (0.67) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
Hydrochloric Acid SCHEMBL989849 0.91 SLC6A9 (0.66) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
SCHEMBL12665683 0.83 SLC6A9 (0.62) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
SCHEMBL8013404 0.83 SLC6A9 (0.73) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
SCHEMBL989105 0.83 SLC6A9 (0.68) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
Hydrochloric Acid SCHEMBL991811 0.82 SLC6A9 (0.72) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
SCHEMBL988895 0.81 SLC6A9 (0.71) SLC6A9CYP3A4MTNR1AMTNR1BNQO2
SCHEMBL8029300 0.79 SLC6A9 (0.63) SLC6A9CYP3A4
SCHEMBL12096285 0.77 SLC6A9 (0.72) SLC6A9CYP3A4
SCHEMBL988862 0.77 SLC6A9 (0.65) SLC6A9CYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2271625-B1 TETRAHYDROISOQUINOLINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE IN THERAPY ABBOTT GMBH & CO KG (DE) 2012-09-12 EP disclosed