SCHEMBL12119908

SCHEMBL12119908

C#CCN[C@@H](C=O)CSCc1ccc(O)c2ncccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.47
MAOB P27338 4/20 0.47
ACHE P22303 1/20 0.47
BACE1 P56817 1/20 0.47
BRD4 O60885 1/20 0.46
KDM4E B2RXH2 7/20 0.44
HTT P42858 4/20 0.44
L3MBTL1 Q9Y468 4/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
LMNA P02545 3/20 0.44
GAA P10253 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALOX12 P18054 3/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALOX15 P16050 3/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
HIF1A Q16665 1/20 0.42
MAPT P10636 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12119911 1.00 MAOA (0.47) MAOAMAOBACHEBACE1BRD4
SCHEMBL113669 0.84 BRD4 (0.48) MAOAMAOBACHEBACE1BRD4
SCHEMBL112274 0.84 BRD4 (0.48) MAOAMAOBACHEBACE1BRD4
SCHEMBL113635 0.84 BRD4 (0.48) MAOAMAOBACHEBACE1BRD4
SCHEMBL12119901 0.78 BRD4 (0.53) BRD4KDM4EHTTL3MBTL1NPC1
SCHEMBL113620 0.74 MAOA (0.53) MAOAMAOBACHEBACE1BRD4
SCHEMBL112261 0.74 MAOA (0.53) MAOAMAOBACHEBACE1BRD4
SCHEMBL113766 0.74 MAOA (0.53) MAOAMAOBACHEBACE1BRD4
SCHEMBL112199 0.74 MAOA (0.80) MAOAMAOBACHEBACE1KDM4E
SCHEMBL12119930 0.72 SLC17A5 (0.44) BRD4KDM4EHTTL3MBTL1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8058442-B2 Neuroprotective iron chelators and pharmaceutical compositions comprising them TECHNION RESEARCH AND DEVELOPMENT FOUNDATION LTD. (IL) 2011-11-15 US disclosed