SCHEMBL12159337

SCHEMBL12159337

C[C@H]1C=Cc2ccccc2N1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.44
MAPT P10636 2/20 0.44
CREBBP Q92793 4/20 0.35
BRPF1 P55201 1/20 0.35
NOS2 P35228 2/20 0.33
BRD4 O60885 4/20 0.32
EP300 Q09472 1/20 0.32
HTR5A P47898 1/20 0.32
P2RX4 Q99571 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
PTPN1 P18031 1/20 0.31
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
GFER P55789 1/20 0.31
TNKS2 Q9H2K2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6056252 1.00 GAA (0.44) GAAMAPTCREBBPBRPF1NOS2
SCHEMBL4705187 0.77 CREBBP (0.38) GAAMAPTCREBBPBRPF1NOS2
SCHEMBL24383177 0.75 NOS2 (0.39) GAAMAPTCREBBPBRPF1NOS2
SCHEMBL4283708 0.74 GAA (0.44) GAAMAPTCREBBPBRPF1BRD4
SCHEMBL5470066 0.74 GAA (0.44) GAAMAPTNOS2
SCHEMBL7442660 0.74 GAA (0.44) GAAMAPTMEN1KMT2AALOX15
SCHEMBL6111309 0.74 GAA (0.44) GAAMAPTCREBBPBRD4P2RX4
SCHEMBL18562457 0.74 GAA (0.44) GAAMAPT
SCHEMBL4540870 0.74 GAA (0.44) GAAMAPT
SCHEMBL13368086 0.74 GAA (0.40) GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2386553-A1 BENZIMIDAZOLE-4-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION METHODS, PHARMACEUTICAL COMPOSITIONS AND THEIR USES Shanghai Jiao Tong University (CN) 2011-11-16 EP disclosed